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#TitleJournalYearCitations
1Dirhodium-catalyzed C-H arene amination using hydroxylaminesScience2016224
2A brief history of antibiotics and select advances in their synthesisJournal of Antibiotics2018121
3Practical access to axially chiral sulfonamides and biaryl amino phenols via organocatalytic atroposelective N-alkylationNature Communications201983
4Total Synthesis and Biological Evaluation of Natural and Designed TubulysinsJournal of the American Chemical Society201678
5The Role of Organic Synthesis in the Emergence and Development of Antibody–Drug Conjugates as Targeted Cancer TherapiesAngewandte Chemie - International Edition201975
6Streamlined Total Synthesis of Uncialamycin and Its Application to the Synthesis of Designed Analogues for Biological InvestigationsJournal of the American Chemical Society201669
7Organic synthesis: the art and science of replicating the molecules of living nature and creating others like them in the laboratoryProceedings of the Royal Society A: Mathematical, Physical and Engineering Sciences201466
8Rapid heteroatom transfer to arylmetals utilizing multifunctional reagent scaffoldsNature Chemistry201763
9Practical Singly and Doubly Electrophilic Aminating Agents: A New, More Sustainable Platform for Carbon–Nitrogen Bond FormationJournal of the American Chemical Society201760
10Total Syntheses of Thailanstatins A–C, Spliceostatin D, and Analogues Thereof. Stereodivergent Synthesis of Tetrasubstituted Dihydro- and Tetrahydropyrans and Design, Synthesis, Biological Evaluation, and Discovery of Potent Antitumor AgentsJournal of the American Chemical Society201845
11Organocatalytic nitrogen transfer to unactivated olefins via transient oxaziridinesNature Catalysis202045
12Improved Total Synthesis of Tubulysins and Design, Synthesis, and Biological Evaluation of New Tubulysins with Highly Potent Cytotoxicities against Cancer Cells as Potential Payloads for Antibody–Drug ConjugatesJournal of the American Chemical Society201844
13Hydrogenation of Alkenes via Cooperative Hydrogen Atom TransferJournal of the American Chemical Society202044
14Total Synthesis of Δ12‐Prostaglandin J3, a Highly Potent and Selective Antileukemic AgentAngewandte Chemie - International Edition201439
15Total Synthesis and Structural Revision of Antibiotic CJ‐16,264Angewandte Chemie - International Edition201539
16Total Synthesis of Trioxacarcins DC-45-A1, A, D, C, and C7″-epi-C and Full Structural Assignment of Trioxacarcin CJournal of the American Chemical Society201639
17Cascade Approach to Highly Functionalized Biaryls by a Nucleophilic Aromatic Substitution with ArylhydroxylaminesOrganic Letters201938
18Total Synthesis and Biological Evaluation of Tiancimycins A and B, Yangpumicin A, and Related Anthraquinone-Fused Enediyne Antitumor AntibioticsJournal of the American Chemical Society202037
19Total Synthesis of Myceliothermophins C, D, and EAngewandte Chemie - International Edition201436
2012,13-Aziridinyl Epothilones. Stereoselective Synthesis of Trisubstituted Olefinic Bonds from Methyl Ketones and Heteroaromatic Phosphonates and Design, Synthesis, and Biological Evaluation of Potent Antitumor AgentsJournal of the American Chemical Society201736
21Streamlined Total Synthesis of Shishijimicin A and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues thereof and Practical Syntheses of PhthNSSMe and Related Sulfenylating ReagentsJournal of the American Chemical Society201836
22Synthesis and Biological Evaluation of QRSTUVWXYZA′ Domains of MaitotoxinJournal of the American Chemical Society201435
23Total Synthesis in Search of Potent Antibody–Drug Conjugate Payloads. From the Fundamentals to the TranslationalAccounts of Chemical Research201934
24Total Synthesis Endeavors and Their Contributions to Science and Society:A Personal AccountCCS Chemistry034
25Synthesis and Biological Investigation of Δ12-Prostaglandin J3 (Δ12-PGJ3) Analogues and Related CompoundsJournal of the American Chemical Society201633
26Total Syntheses of Disorazoles A1 and B1 and Full Structural Elucidation of Disorazole B1Journal of the American Chemical Society201733
27The Emergence and Evolution of Organic Synthesis and Why It is Important to Sustain It as an Advancing Art and Science for Its Own SakeIsrael Journal of Chemistry201833
28Recent Advances in Small Molecule‐Based Intracellular pH ProbesChemBioChem202230
29Total Synthesis of Trioxacarcin DC‐45‐A2Angewandte Chemie - International Edition201523
30Total Synthesis of Δ12‐Prostaglandin J3: Evolution of Synthetic Strategies to a Streamlined ProcessChemistry - A European Journal201622
31Practical Synthesis of p‐ and o‐Amino‐ and Methoxyphenolic AnthraquinonesAngewandte Chemie - International Edition201520
32DNA Binding and Cleavage Modes of Shishijimicin AJournal of the American Chemical Society201920
33Uncialamycin-based antibody–drug conjugates: Unique enediyne ADCs exhibiting bystander killing effectProceedings of the National Academy of Sciences of the United States of America202120
34The Chemistry-Biology-Medicine Continuum and the Drug Discovery and Development Process in AcademiaChemistry and Biology201419
35Total Synthesis and Full Structural Assignment of NamenamicinJournal of the American Chemical Society201818
36Total Synthesis of the Monomeric Unit of Lomaiviticin AJournal of the American Chemical Society202018
37Catalyst: Synthetic Organic Chemistry as a Force for GoodCheM201617
38Design, Synthesis, and Biological Investigation of Epothilone B Analogues Featuring Lactone, Lactam, and Carbocyclic Macrocycles, Epoxide, Aziridine, and 1,1-Difluorocyclopropane and Other Fluorine ResiduesJournal of Organic Chemistry202017
39A Reverse Approach to the Total Synthesis of Halichondrin BJournal of the American Chemical Society202116
40Cyclopamine analogs bearing exocyclic methylenes are highly potent and acid-stable inhibitors of hedgehog signalingBeilstein Journal of Organic Chemistry201315
41Short Total Synthesis of Δ12-Prostaglandin J2 and Related Prostaglandins. Design, Synthesis, and Biological Evaluation of Macrocyclic Δ12-Prostaglandin J2 AnaloguesJournal of Organic Chemistry201915
42Streamlined Total Synthesis of Trioxacarcins and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues Thereof. Discovery of Simpler Designed and Potent Trioxacarcin AnaloguesJournal of the American Chemical Society201714
43Transition metal-free direct dehydrogenative arylation of activated C(sp3)–H bonds: synthetic ambit and DFT reactivity predictionsChemical Science201814
44Streamlined Symmetrical Total Synthesis of Disorazole B1 and Design, Synthesis, and Biological Investigation of Disorazole AnaloguesJournal of the American Chemical Society202014
45Syntheses of Cyclopropyl Analogues of Disorazoles A1 and B1 and Their Thiazole CounterpartsJournal of Organic Chemistry201813
46Overview of Amino Acid Modifications by Iron- and α-Ketoglutarate-Dependent EnzymesACS Catalysis202312
47C–H-Functionalization logic guides the synthesis of a carbacyclopamine analogBeilstein Journal of Organic Chemistry201411
48Efficient Synthesis of Dimeric Oxazoles, Piperidines and Tetrahydroisoquinolines from N‐Substituted 2‐OxazolonesChemistry - A European Journal201611
49Die Bedeutung der organischen Synthese bei der Entstehung und Entwicklung von Antikörper‐Wirkstoff‐Konjugaten als gezielte KrebstherapienAngewandte Chemie201911
50Synthesis and Biological Evaluation of Shishijimicin A-Type Linker-Drugs and Antibody–Drug ConjugatesJournal of the American Chemical Society202011